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Description

Notopterol mitigates osteoarthritis progression and relieves pain in mice by inhibiting PI3K/Akt/GPX4-mediated ferroptosis

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In addition to stimulating calcium overload caused by ATP enzyme imbalances, such as imbalances in calcium pump activity, metabolites, including lactic acid and succinic acid, accumulate, antioxidant enzyme activity is inhibited, the mitochondrial structure is destroyed and mitochondrial function is dysregulated under ischemic conditions

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Oral forms exist but have lower absorption

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GeroScience 44 , 26232653 (2022)

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